F2RL1
F2R like trypsin receptor 1 | PAR2, GPR11

This gene encodes a member of the G-protein coupled receptor 1 family of proteins. The encoded cell surface receptor is activated through proteolytic cleavage of its extracellular amino terminus, resulting in a new amino terminus that acts as a tethered ligand that binds to an extracellular loop domain. Activation of the receptor has been shown to stimulate vascular smooth muscle relaxation, dilate blood vessels, increase blood flow, and lower blood pressure. This protein is also important in the inflammatory response, as well as innate and adaptive immunity. [provided by RefSeq, Jun 2016]

Developmental clusters: GC4
Biological processes 99 terms
G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor signaling pathway (GO:0007186)G protein-coupled receptor signaling pathway (GO:0007186)G protein-coupled receptor signaling pathway (GO:0007186)G protein-coupled receptor signaling pathway (GO:0007186)G-protein alpha-subunit binding (GO:0001965)G-protein alpha-subunit binding (GO:0001965)G-protein beta-subunit binding (GO:0031681)G-protein beta-subunit binding (GO:0031681)Golgi apparatus (GO:0005794)T cell activation involved in immune response (GO:0002286)T cell activation involved in immune response (GO:0002286)antimicrobial humoral response (GO:0019730)blood coagulation (GO:0007596)cell-cell junction maintenance (GO:0045217)defense response to virus (GO:0051607)defense response to virus (GO:0051607)early endosome (GO:0005769)establishment of endothelial barrier (GO:0061028)leukocyte migration (GO:0050900)leukocyte proliferation (GO:0070661)leukocyte proliferation (GO:0070661)mature conventional dendritic cell differentiation (GO:0097029)mature conventional dendritic cell differentiation (GO:0097029)mature conventional dendritic cell differentiation (GO:0097029)membrane (GO:0016020)negative regulation of JNK cascade (GO:0046329)negative regulation of chemokine production (GO:0032682)negative regulation of toll-like receptor 3 signaling pathway (GO:0034140)negative regulation of tumor necrosis factor-mediated signaling pathway (GO:0010804)neutrophil activation (GO:0042119)plasma membrane (GO:0005886)plasma membrane (GO:0005886)plasma membrane (GO:0005886)plasma membrane (GO:0005886)positive regulation of ERK1 and ERK2 cascade (GO:0070374)positive regulation of ERK1 and ERK2 cascade (GO:0070374)positive regulation of ERK1 and ERK2 cascade (GO:0070374)positive regulation of ERK1 and ERK2 cascade (GO:0070374)positive regulation of JNK cascade (GO:0046330)positive regulation of Rho protein signal transduction (GO:0035025)positive regulation of Rho protein signal transduction (GO:0035025)positive regulation of Rho protein signal transduction (GO:0035025)positive regulation of Rho protein signal transduction (GO:0035025)positive regulation of actin filament depolymerization (GO:0030836)positive regulation of canonical NF-kappaB signal transduction (GO:0043123)positive regulation of cell migration (GO:0030335)positive regulation of cell migration (GO:0030335)positive regulation of chemokine production (GO:0032722)positive regulation of chemokine production (GO:0032722)positive regulation of chemotaxis (GO:0050921)positive regulation of chemotaxis (GO:0050921)positive regulation of cytokine production involved in immune response (GO:0002720)positive regulation of cytosolic calcium ion concentration (GO:0007204)positive regulation of cytosolic calcium ion concentration (GO:0007204)positive regulation of cytosolic calcium ion concentration (GO:0007204)positive regulation of cytosolic calcium ion concentration (GO:0007204)positive regulation of eosinophil degranulation (GO:0043311)positive regulation of glomerular filtration (GO:0003104)positive regulation of glomerular filtration (GO:0003104)positive regulation of interleukin-1 beta production (GO:0032731)positive regulation of interleukin-10 production (GO:0032733)positive regulation of interleukin-6 production (GO:0032755)positive regulation of interleukin-8 production (GO:0032757)positive regulation of leukocyte chemotaxis (GO:0002690)positive regulation of phagocytosis, engulfment (GO:0060100)positive regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction (GO:0051897)positive regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction (GO:0051897)positive regulation of positive chemotaxis (GO:0050927)positive regulation of pseudopodium assembly (GO:0031274)positive regulation of pseudopodium assembly (GO:0031274)positive regulation of renin secretion into blood stream (GO:1900135)positive regulation of renin secretion into blood stream (GO:1900135)positive regulation of superoxide anion generation (GO:0032930)positive regulation of toll-like receptor 2 signaling pathway (GO:0034137)positive regulation of toll-like receptor 3 signaling pathway (GO:0034141)positive regulation of toll-like receptor 4 signaling pathway (GO:0034145)positive regulation of transcription by RNA polymerase II (GO:0045944)positive regulation of type II interferon production (GO:0032729)positive regulation of type II interferon production (GO:0032729)protease binding (GO:0002020)protein binding (GO:0005515)proteinase-activated receptor activity (GO:0001648)pseudopodium (GO:0031143)pseudopodium (GO:0031143)regulation of JNK cascade (GO:0046328)regulation of blood coagulation (GO:0030193)regulation of canonical NF-kappaB signal transduction (GO:0043122)regulation of chemokine (C-X-C motif) ligand 2 production (GO:2000341)signaling receptor activity (GO:0038023)signaling receptor binding (GO:0005102)thrombin-activated receptor activity (GO:0015057)thrombin-activated receptor signaling pathway (GO:0070493)vasodilation (GO:0042311)vasodilation (GO:0042311)
Expression (TPM)
F2RL1 — as a Regulated Gene

TFs regulating F2RL1 0 TFs

Transcription factors with Perturb-seq knockdown data for F2RL1. The Binding column indicates whether any binding evidence exists for this TF–gene pair (ChIP-seq or motif footprint peaks). The Mean coef is the average Perturb-seq regression coefficient across active gRNAs (positive = F2RL1 upregulated upon KD; negative = downregulated). The Outlier column indicates whether this gene is in the top or bottom 5% of all TF knockdown effects.

Data: Effect:
TF Mean coef Binding Outlier TF→Gene link

Elements linked to F2RL1

Open chromatin peaks (ATAC-seq) in the genomic neighbourhood of F2RL1, linked by TSS proximity or chromatin conformation (Multiome / HiCAR). Each element overlaps at least one TF ChIP-seq binding site — the TFs column shows how many distinct TFs bind that element.

Accessibility Element Dist. to TSS Link type TFs
chr5:76,548,249–76,549,423 270.3 kb Distal (>10kb) Multiome 149
chr5:76,715,026–76,716,740 103.0 kb Distal (>10kb) Multiome 666
chr5:76,789,270–76,790,249 29.1 kb Distal (>10kb) Multiome 123
chr5:76,808,093–76,808,802 10.6 kb Distal (>10kb) Multiome 237
chr5:76,809,142–76,809,507 9.5 kb Proximal (<10kb) 39
chr5:76,818,219–76,818,362 666 bp At TSS 36
chr5:76,818,476–76,819,940 71 bp At TSS Multiome 686
chr5:76,820,052–76,820,315 1.0 kb Proximal (<10kb) 228
chr5:76,821,065–76,821,450 2.0 kb Proximal (<10kb) 37
chr5:76,873,943–76,874,791 55.4 kb Distal (>10kb) Multiome 261
chr5:76,953,306–76,954,445 134.7 kb Distal (>10kb) Multiome 235
chr5:77,030,193–77,031,058 211.4 kb Distal (>10kb) Multiome 903
chr5:77,076,843–77,078,059 258.6 kb Distal (>10kb) Multiome 396
chr5:77,086,556–77,087,540 267.9 kb Distal (>10kb) Multiome 768

Genome Browser

Genomic view of the F2RL1 locus showing ATAC-seq accessibility and RNA-seq expression across the ESC → DE time course, together with TF binding peaks and element-to-TSS loop connections.

chr5:76,538,249 – 77,097,540
Proximal 1 kb Distal 10 kb Multiome HiCAR ATAC-seq RNA-seq