F2R
coagulation factor II thrombin receptor | CF2R, PAR-1, PAR1, TR

Coagulation factor II receptor is a 7-transmembrane receptor involved in the regulation of thrombotic response. Proteolytic cleavage leads to the activation of the receptor. F2R is a G-protein coupled receptor family member. Alternative splicing results in multiple transcript variants. [provided by RefSeq, Aug 2015]

Member of: DE-3 DE-3.50
Biological processes 83 terms
G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor activity (GO:0004930)G protein-coupled receptor signaling pathway (GO:0007186)G protein-coupled receptor signaling pathway (GO:0007186)G-protein alpha-subunit binding (GO:0001965)G-protein alpha-subunit binding (GO:0001965)G-protein beta-subunit binding (GO:0031681)G-protein beta-subunit binding (GO:0031681)Golgi apparatus (GO:0005794)anatomical structure morphogenesis (GO:0009653)blood coagulation (GO:0007596)caveola (GO:0005901)cell surface (GO:0009986)cell-cell junction maintenance (GO:0045217)connective tissue replacement involved in inflammatory response wound healing (GO:0002248)early endosome (GO:0005769)establishment of synaptic specificity at neuromuscular junction (GO:0007529)extracellular region (GO:0005576)homeostasis of number of cells within a tissue (GO:0048873)inflammatory response (GO:0006954)late endosome (GO:0005770)membrane (GO:0016020)negative regulation of cell population proliferation (GO:0008285)negative regulation of glomerular filtration (GO:0003105)negative regulation of neuron apoptotic process (GO:0043524)negative regulation of renin secretion into blood stream (GO:1900134)negative regulation of renin secretion into blood stream (GO:1900134)neuromuscular junction (GO:0031594)phospholipase C-activating G protein-coupled receptor signaling pathway (GO:0007200)phospholipase C-activating G protein-coupled receptor signaling pathway (GO:0007200)phospholipase C-activating G protein-coupled receptor signaling pathway (GO:0007200)plasma membrane (GO:0005886)plasma membrane (GO:0005886)plasma membrane (GO:0005886)plasma membrane (GO:0005886)plasma membrane (GO:0005886)platelet activation (GO:0030168)platelet dense granule organization (GO:0060155)platelet dense tubular network (GO:0031094)positive regulation of DNA-templated transcription (GO:0045893)positive regulation of ERK1 and ERK2 cascade (GO:0070374)positive regulation of ERK1 and ERK2 cascade (GO:0070374)positive regulation of MAPK cascade (GO:0043410)positive regulation of Rho protein signal transduction (GO:0035025)positive regulation of Rho protein signal transduction (GO:0035025)positive regulation of apoptotic process (GO:0043065)positive regulation of blood coagulation (GO:0030194)positive regulation of blood coagulation (GO:0030194)positive regulation of calcium ion transport (GO:0051928)positive regulation of canonical NF-kappaB signal transduction (GO:0043123)positive regulation of cell migration (GO:0030335)positive regulation of cell migration (GO:0030335)positive regulation of cell population proliferation (GO:0008284)positive regulation of collagen biosynthetic process (GO:0032967)positive regulation of cytosolic calcium ion concentration (GO:0007204)positive regulation of cytosolic calcium ion concentration (GO:0007204)positive regulation of interleukin-6 production (GO:0032755)positive regulation of interleukin-8 production (GO:0032757)positive regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction (GO:0051897)positive regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction (GO:0051897)positive regulation of receptor signaling pathway via JAK-STAT (GO:0046427)positive regulation of release of sequestered calcium ion into cytosol (GO:0051281)positive regulation of smooth muscle contraction (GO:0045987)positive regulation of vasoconstriction (GO:0045907)positive regulation of vasoconstriction (GO:0045907)postsynaptic membrane (GO:0045211)protein binding (GO:0005515)regulation of blood coagulation (GO:0030193)regulation of interleukin-1 beta production (GO:0032651)regulation of synaptic plasticity (GO:0048167)regulation of synaptic plasticity (GO:0048167)release of sequestered calcium ion into cytosol (GO:0051209)response to lipopolysaccharide (GO:0032496)response to wounding (GO:0009611)signaling receptor binding (GO:0005102)thrombin-activated receptor activity (GO:0015057)thrombin-activated receptor activity (GO:0015057)thrombin-activated receptor activity (GO:0015057)thrombin-activated receptor activity (GO:0015057)thrombin-activated receptor signaling pathway (GO:0070493)thrombin-activated receptor signaling pathway (GO:0070493)trans-synaptic signaling by endocannabinoid, modulating synaptic transmission (GO:0099553)
Expression (TPM)
F2R — as a Regulated Gene

TFs regulating F2R 0 TFs

Transcription factors with Perturb-seq knockdown data for F2R. The Binding column indicates whether any binding evidence exists for this TF–gene pair (ChIP-seq or motif footprint peaks). The Mean coef is the average Perturb-seq regression coefficient across active gRNAs (positive = F2R upregulated upon KD; negative = downregulated). The Outlier column indicates whether this gene is in the top or bottom 5% of all TF knockdown effects.

Data: Effect:
TF Mean coef Binding Outlier TF→Gene link

Elements linked to F2R

Open chromatin peaks (ATAC-seq) in the genomic neighbourhood of F2R, linked by TSS proximity or chromatin conformation (Multiome / HiCAR). Each element overlaps at least one TF ChIP-seq binding site — the TFs column shows how many distinct TFs bind that element.

Accessibility Element Dist. to TSS Link type TFs
chr5:76,504,460–76,505,155 211.3 kb Distal (>10kb) Multiome 40
chr5:76,548,249–76,549,423 167.4 kb Distal (>10kb) Multiome 149
chr5:76,715,026–76,716,740 54 bp At TSS Multiome 666
chr5:76,716,876–76,717,040 751 bp At TSS 180
chr5:76,789,270–76,790,249 73.8 kb Distal (>10kb) Multiome 123
chr5:76,808,093–76,808,802 92.3 kb Distal (>10kb) Multiome 237
chr5:76,818,476–76,819,940 102.8 kb Distal (>10kb) Multiome 686
chr5:76,873,943–76,874,791 158.3 kb Distal (>10kb) Multiome 261
chr5:76,953,306–76,954,445 237.6 kb Distal (>10kb) Multiome 235

Genome Browser

Genomic view of the F2R locus showing ATAC-seq accessibility and RNA-seq expression across the ESC → DE time course, together with TF binding peaks and element-to-TSS loop connections.

chr5:76,494,460 – 76,964,445
Proximal 1 kb Distal 10 kb Multiome HiCAR ATAC-seq RNA-seq