PDK2
pyruvate dehydrogenase kinase 2 | PDHK2

This gene encodes a member of the pyruvate dehydrogenase kinase family. The encoded protein phosphorylates pyruvate dehydrogenase, down-regulating the activity of the mitochondrial pyruvate dehydrogenase complex. Overexpression of this gene may play a role in both cancer and diabetes. Alternatively spliced transcript variants encoding multiple isoforms have been observed for this gene. [provided by RefSeq, Dec 2010]

Biological processes 39 terms
ATP binding (GO:0005524)cellular response to nutrient (GO:0031670)cellular response to nutrient (GO:0031670)cellular response to reactive oxygen species (GO:0034614)cellular response to stress (GO:0033554)glucose homeostasis (GO:0042593)glucose homeostasis (GO:0042593)glucose metabolic process (GO:0006006)insulin receptor signaling pathway (GO:0008286)insulin receptor signaling pathway (GO:0008286)intrinsic apoptotic signaling pathway by p53 class mediator (GO:0072332)mitochondrial matrix (GO:0005759)mitochondrial matrix (GO:0005759)mitochondrion (GO:0005739)mitochondrion (GO:0005739)mitochondrion (GO:0005739)mitochondrion (GO:0005739)protein binding (GO:0005515)protein homodimerization activity (GO:0042803)protein kinase activity (GO:0004672)protein kinase activity (GO:0004672)pyruvate dehydrogenase (acetyl-transferring) kinase activity (GO:0004740)pyruvate dehydrogenase (acetyl-transferring) kinase activity (GO:0004740)pyruvate dehydrogenase (acetyl-transferring) kinase activity (GO:0004740)pyruvate dehydrogenase (acetyl-transferring) kinase activity (GO:0004740)pyruvate dehydrogenase complex (GO:0045254)pyruvate dehydrogenase complex (GO:0045254)regulation of gluconeogenesis (GO:0006111)regulation of gluconeogenesis (GO:0006111)regulation of glucose metabolic process (GO:0010906)regulation of glucose metabolic process (GO:0010906)regulation of glucose metabolic process (GO:0010906)regulation of ketone metabolic process (GO:0010565)regulation of ketone metabolic process (GO:0010565)regulation of pH (GO:0006885)regulation of pH (GO:0006885)regulation of pyruvate decarboxylation to acetyl-CoA (GO:0010510)regulation of pyruvate decarboxylation to acetyl-CoA (GO:0010510)regulation of pyruvate decarboxylation to acetyl-CoA (GO:0010510)
Expression (TPM)
PDK2 — as a Regulated Gene

TFs regulating PDK2 0 TFs

Transcription factors with Perturb-seq knockdown data for PDK2. The Binding column indicates whether any binding evidence exists for this TF–gene pair (ChIP-seq or motif footprint peaks). The Mean coef is the average Perturb-seq regression coefficient across active gRNAs (positive = PDK2 upregulated upon KD; negative = downregulated). The Outlier column indicates whether this gene is in the top or bottom 5% of all TF knockdown effects.

Data: Effect:
TF Mean coef Binding Outlier TF→Gene link

Elements linked to PDK2

Open chromatin peaks (ATAC-seq) in the genomic neighbourhood of PDK2, linked by TSS proximity or chromatin conformation (Multiome / HiCAR). Each element overlaps at least one TF ChIP-seq binding site — the TFs column shows how many distinct TFs bind that element.

Accessibility Element Dist. to TSS Link type TFs
chr17:50,087,492–50,087,764 7.6 kb Proximal (<10kb) 384
chr17:50,094,331–50,095,951 at TSS At TSS 899

Genome Browser

Genomic view of the PDK2 locus showing ATAC-seq accessibility and RNA-seq expression across the ESC → DE time course, together with TF binding peaks and element-to-TSS loop connections.

chr17:50,077,492 – 50,105,951
Proximal 1 kb Distal 10 kb Multiome HiCAR ATAC-seq RNA-seq