PDE3A
phosphodiesterase 3A | CGI-PDE

This gene encodes a member of the cGMP-inhibited cyclic nucleotide phosphodiesterase (cGI-PDE) family. cGI-PDE enzymes hydrolyze both cAMP and cGMP, and play critical roles in many cellular processes by regulating the amplitude and duration of intracellular cyclic nucleotide signals. The encoded protein mediates platelet aggregation and also plays important roles in cardiovascular function by regulating vascular smooth muscle contraction and relaxation. Inhibitors of the encoded protein may be effective in treating congestive heart failure. Alternatively spliced transcript variants encoding multiple isoforms have been observed for this gene. [provided by RefSeq, Sep 2011]

Biological processes 37 terms
3',5'-cGMP-inhibited cyclic-nucleotide phosphodiesterase activity (GO:0004119)3',5'-cGMP-inhibited cyclic-nucleotide phosphodiesterase activity (GO:0004119)3',5'-cyclic-AMP phosphodiesterase activity (GO:0004115)3',5'-cyclic-AMP phosphodiesterase activity (GO:0004115)3',5'-cyclic-AMP phosphodiesterase activity (GO:0004115)3',5'-cyclic-AMP phosphodiesterase activity (GO:0004115)3',5'-cyclic-GMP phosphodiesterase activity (GO:0047555)3',5'-cyclic-GMP phosphodiesterase activity (GO:0047555)3',5'-cyclic-GMP phosphodiesterase activity (GO:0047555)3',5'-cyclic-nucleotide phosphodiesterase activity (GO:0004114)3',5'-cyclic-nucleotide phosphodiesterase activity (GO:0004114)G protein-coupled receptor signaling pathway (GO:0007186)apoptotic signaling pathway (GO:0097190)cellular response to cGMP (GO:0071321)cellular response to transforming growth factor beta stimulus (GO:0071560)cytosol (GO:0005829)cytosol (GO:0005829)cytosol (GO:0005829)cytosol (GO:0005829)estrogen binding (GO:0099130)lipid metabolic process (GO:0006629)membrane (GO:0016020)negative regulation of adenylate cyclase-activating G protein-coupled receptor signaling pathway (GO:0106072)negative regulation of adenylate cyclase-activating G protein-coupled receptor signaling pathway (GO:0106072)negative regulation of apoptotic process (GO:0043066)negative regulation of cAMP/PKA signal transduction (GO:0141162)negative regulation of cAMP/PKA signal transduction (GO:0141162)negative regulation of vascular permeability (GO:0043116)nuclear estrogen receptor activity (GO:0030284)nuclear receptor-mediated steroid hormone signaling pathway (GO:0030518)oocyte maturation (GO:0001556)phosphoric diester hydrolase activity (GO:0008081)positive regulation of vascular permeability (GO:0043117)protein binding (GO:0005515)regulation of ribonuclease activity (GO:0060700)regulation of ribonuclease activity (GO:0060700)signal transduction (GO:0007165)
Expression (TPM)
PDE3A — as a Regulated Gene

TFs regulating PDE3A 0 TFs

Transcription factors with Perturb-seq knockdown data for PDE3A. The Binding column indicates whether any binding evidence exists for this TF–gene pair (ChIP-seq or motif footprint peaks). The Mean coef is the average Perturb-seq regression coefficient across active gRNAs (positive = PDE3A upregulated upon KD; negative = downregulated). The Outlier column indicates whether this gene is in the top or bottom 5% of all TF knockdown effects.

Data: Effect:
TF Mean coef Binding Outlier TF→Gene link

Elements linked to PDE3A

Open chromatin peaks (ATAC-seq) in the genomic neighbourhood of PDE3A, linked by TSS proximity or chromatin conformation (Multiome / HiCAR). Each element overlaps at least one TF ChIP-seq binding site — the TFs column shows how many distinct TFs bind that element.

Accessibility Element Dist. to TSS Link type TFs
chr12:20,212,609–20,213,324 155.6 kb Distal (>10kb) Multiome 392
chr12:20,264,125–20,265,112 103.8 kb Distal (>10kb) Multiome 206
chr12:20,367,802–20,370,591 1.2 kb Proximal (<10kb) Multiome 513

Genome Browser

Genomic view of the PDE3A locus showing ATAC-seq accessibility and RNA-seq expression across the ESC → DE time course, together with TF binding peaks and element-to-TSS loop connections.

chr12:20,202,609 – 20,380,591
Proximal 1 kb Distal 10 kb Multiome HiCAR ATAC-seq RNA-seq